| Strategies toward Dicarbofunctionalization of Unactivated Olefins by Combined Heck Carbometalation and Cross-Coupling |
59 |
| Sustainability Challenges in Peptide Synthesis and Purification: From R&D to Production |
45 |
| Visible Light-Induced Thiocyanation of Enaminone C-H Bond to Access Polyfunctionalized Alkenes and Thiocyano Chromones |
39 |
| En Route to Intermolecular Cross-Dehydrogenative Coupling Reactions |
36 |
| Iodine-Mediated Difunctionalization of Imidazopyridines with Sodium Sulfinates: Synthesis of Sulfones and Sulfides |
34 |
| Asymmetric Synthesis of Dihydrocoumarins through Chiral Phosphoric Acid-Catalyzed Cycloannulation of para-Quinone Methides and Azlactones |
30 |
| Selective Synthesis of 2-Substituted and 2-Disubstituted Benzimidazoles Directly from Aromatic Diamines and Alcohols Catalyzed by Molecularly Defined Nonphosphine Manganese(I) Complex |
28 |
| Iodine-Catalyzed Odorless Synthesis of S-Thiocarbamates with Sulfonyl Chlorides as a Sulfur Source |
26 |
| Catalytic Asymmetric [4+1] Cyclization of Benzofuran-Derived Azadienes with 3-Chlorooxindoles |
25 |
| Absolute Configurations of Synthetic Molecular Scaffolds from Vibrational CD Spectroscopy |
24 |
| Synthesis of Polysubstituted Quinolines from alpha-2-Aminoaryl Alcohols Via Nickel-Catalyzed Dehydrogenative Coupling |
24 |
| Domino C-H Sulfonylation and Pyrazole Annulation for Fully Substituted Pyrazole Synthesis in Water Using Hydrophilic Enaminones |
23 |
| Organocatalyzed, Visible-Light Photoredox-Mediated, One-Pot Minisci Reaction Using Carboxylic Acids via N-(Acyloxy)phthalimides |
23 |
| Metal-Catalyzed Oxa-[4+2] Cyclizations of Quinone Methides with Alkynyl Benzyl Alcohols |
23 |
| [3+2]-Cycloaddition of in Situ Generated Nitrile lmines and Acetylene for Assembling of 3-Disubstituted Pyrazoles with Quantitative Deuterium Labeling |
23 |
| Enantioselective N-Heterocyclic Carbene-Catalyzed Synthesis of Spirocyclic Oxindole-benzofuroazepinones |
23 |
| Asymmetric Rhodium-Catalyzed Allylic Substitution Reactions: Discovery, Development and Applications to Target-Directed Synthesis |
22 |
| Tunable Synthesis of 3-Hydroxylisoquinolin-4-dione and Isoquinolin-1-one Enabled by Copper-Catalyzed Radical 6-endo Aza-cyclization of 2-Alkynylbenzamide |
21 |
| Copper-Mediated C-H Amination of Imidazopyridines with N-Fluorobenzenesulfonimide |
21 |
| Regioselective Halogenation of Arenes and Heterocycles in Hexafluoroisopropanol |
21 |
| A Molecular Electron Density Theory Study of the Reactivity and Selectivities in [3+2] Cycloaddition Reactions of C,N-Dialkyl Nitrones with Ethylene Derivatives |
21 |
| Sodium Salts (NaI/NaBr/NaCl) for the Halogenation of Imidazo-Fused Heterocycles |
21 |
| [4+2] Cyclization of para-Quinone Methide Derivatives with Alkynes |
20 |
| Redesigning the Coumarin Scaffold into Small Bright Fluorophores with Far-Red to Near-Infrared Emission and Large Stokes Shifts Useful for Cell Imaging |
20 |
| Visible Light Induced Metal-Free Carbene N-Carbazolation |
20 |
| Visible-Light-Induced Organophotoredox-Catalyzed Phosphonylation of 2H-Indazoles with Diphenylphosphine Oxide |
20 |
| Insights into N-Heterocyclic Carbene-Catalyzed Oxidative alpha-C(sp(3))-H Activation of Aliphatic Aldehydes and Cascade [2+2] Cycloaddition with Ketimines |
20 |
| Generation of 3-Dimethylene-Substituted Isobenzofurans via Pd(II)-Catalyzed Selective Oxo-cyclization/SO2 Insertion Cascade of beta-Alkynyl Ketones |
19 |
| Tandem Flavin-Iodine-Catalyzed Aerobic Oxidative Sulfenylation of Imidazo[2-a]Pyridines with Thiols |
18 |
| Electron Donor-Acceptor Complex Enabled Decarboxylative Sulfonylation of Cinnamic Acids under Visible-Light Irradiation |
18 |
| Rapidly Activating Pd-Precatalyst for Suzuki-Miyaura and Buchwald-Hartwig Couplings of Aryl Esters |
18 |
| Asymmetric Construction of Bispiro[oxindole-pyrrolidine-rhodanine]s via Squaramide-Catalyzed Domino Michael/Mannich [3+2] Cycloaddition of Rhodanine Derivatives with N-(2-Trifluoroethyl)isatin Ketimines |
18 |
| Application of Naphthylindole-Derived Phosphines as Organocatalysts in [4+1] Cyclizations of o-Quinone Methides with Morita-Baylis-Hillman Carbonates |
18 |
| Three-Component Coupling of Aldehydes, Aminopyrazoles, and Sulfoxonium Ylides via Rhodium(III)-Catalyzed Imidoyl C-H Activation: Synthesis of Pyrazolo[5-a]pyrimidines |
18 |
| Halo-3-triazolium Salts as Halogen Bond Donors for the Activation of Imines in Dihydropyridinone Synthesis |
18 |
| Difluoro-Substituted Bicyclo[1.1.1]pentanes for Medicinal Chemistry: Design, Synthesis, and Characterization |
17 |
| Direct C-H Methylsulfonylation of Alkenes with the Insertion of Sulfur Dioxide |
17 |
| Rh/O-2-Catalyzed C8 Olefination of Quinoline N-Oxides with Activated and Unactivated Olefins |
17 |
| Synthesis of Nitriles from Primary Amides or Aldoximes under Conditions of a Catalytic Swern Oxidation |
17 |
| Organocatalytic Asymmetric Sequential 6-Addition/Acetalization of 1-Oxotetralin-2-carbaldehyde to ortho-Hydroxyphenyl-Substituted para-Quinone Methides for Synthesis of Spiro-4-dihydrocoumarins |
17 |
| Pd-Catalyzed Asymmetric Dearomative Cycloaddition for Construction of Optically Active Pyrroloindoline and Cyclopentaindoline Derivatives: Access to 3a-Aminopyrroloindolines |
17 |
| Direct C3 Alkoxylation of Quinoxalin-2(1H)-ones with Alcohols via Cross-Dehydrogenative Coupling under Catalyst-Free Conditions |
17 |
| Lactam Hydrogen Bonds as Control Elements in Enantioselective Transition-Metal-Catalyzed and Photochemical Reactions |
17 |
| Aromatization-Driven Cascade [5]-Hydride Transfer/Spirocyclization Promoted by Fluorinated Alcohols |
17 |
| Ytterbium-Catalyzed Hydroboration of Aldehydes and Ketones |
17 |
| Insights into the N-Heterocyclic Carbene (NHC)-Catalyzed Oxidative gamma-C(sp(3)) H Deprotonation of Alkylenals and Cascade [4+2] Cycloaddition with Alkenylisoxazoles |
17 |
| Synthesis of (2H)-Indazoles through Rh(III)-Catalyzed Annulation Reaction of Azobenzenes with Sulfoxonium Ylides |
17 |
| Sustainable Alkylation of Nitriles with Alcohols by Manganese Catalysis |
17 |
| Diastereoselective Construction of Indole-Bridged Chroman Spirooxindoles through a TfOH-Catalyzed Michael Addition-Inspired Cascade Reaction |
17 |
| Bioactive Penicipyrrodiether A, an Adduct of GKK1032 Analogue and Phenol A Derivative, from a Marine-Sourced Fungus Penicillium sp ZZ380 |
17 |
