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2H-pyrazolo[3,4-d]pyrimidin-4-amine derivatives as novel selective fibroblast growth factor receptor 2 (FGFR2) inhibitor
Author: Wu, Pinglian; Tian, Zhaodi; Shen, Weizhong; Xun, Qiuju; Tian, Yuan; Li, Huiqiong; Yang, Bowen; Chang, Shaohua; Huang, Weixue; Wang, Zhen; Ding, Ke; Ma, Dawei
Journal: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. 2026; Vol. 41, Issue 1, pp. -. DOI: 10.1080/14756366.2026.2647526
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Application of 18β-glycyrrhetinic acid Fluorescent probes in cell imagin
Author: Zhao, Yifan; Sun, Hongxia; Yan, Zhiwei; Wang, Youde; Li, Shuai; Guo, Yachun; Miao, Guangxin; Wang, Tienan; Zhang, Liying; Song, Chengjun
Journal: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. 2026; Vol. 41, Issue 1, pp. -. DOI: 10.1080/14756366.2026.2631869
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Screening of peptide inhibitors targeting YAP-TEAD4 interaction: affinity evaluation and anti-AML cell activit
Author: Yang, Xiaotian; Yang, Shudan; Lin, Guoqiang; Chen, Shutong; Jiang, Huiran; Wang, Yuting; Zhang, Yanming; Zhang, Xingxia
Journal: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. 2026; Vol. 41, Issue 1, pp. -. DOI: 10.1080/14756366.2026.2633822
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LDH isozymes as targets for cancer therap
Author: Hou, Yiqian; Zhao, Yanying; He, Qinghua; Wang, Meilin; Zhang, Qinglian
Journal: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. 2026; Vol. 41, Issue 1, pp. -. DOI: 10.1080/14756366.2026.2639168
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Drug-likeness prioritised selection identifies anti-Escherichia coli candidates confirmed by molecular docking, dynamics simulations, and antibacterial assay
Author: Yu, Beibei; Zhu, Haoyu; Xu, Lu; Zhao, Xiangdong; Shi, Wei
Journal: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. 2026; Vol. 41, Issue 1, pp. -. DOI: 10.1080/14756366.2026.2640719
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Discovery of ferulic acid carbamate derivatives as dual-targeting agents of BuChE and Nrf2 for Alzheimer's diseas
Author: Lao, Kejing; Li, Yingze; Xiao, Yueyan; Sun, Ya; Dai, Yuxuan; Li, Huijin; Yang, Yang; Zhang, Yun; Wang, Jing; Li, Weize; Gou, Xingchun; Guan, Li
Journal: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. 2026; Vol. 41, Issue 1, pp. -. DOI: 10.1080/14756366.2026.2645483
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Design, synthesis and biological evaluation of donepezil-safinamide hybrids as dual AChE and MAO-B inhibitor for Alzheimer's disease treatmen
Author: Li, Wei; Guo, Yan; Wang, Xiaoli; Yang, Chunyan; Zhu, Jiang; Cao, Zhongcheng
Journal: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. 2026; Vol. 41, Issue 1, pp. -. DOI: 10.1080/14756366.2026.2622769
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Thymol carbamates bearing cyclic amines as potent and selective BuChE inhibitors alleviate memory impairments for Alzheimer's disease therap
Author: Wu, Chengyao; Ding, Yulu; Liu, Xiaodan; Gao, Shan; Wang, Xiaoqing; Tang, Wenjian
Journal: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. 2026; Vol. 41, Issue 1, pp. -. DOI: 10.1080/14756366.2026.2623314