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Synthesis, cytotoxicity, and pharmacokinetic evaluations of niclosamide analogs for anti-SARS-CoV-2
Author: Li, Rui; Zhang, Zherui; Huang, Shuhong; Peng, Ke; Jiang, Hualiang; Shen, Jingshan; Zhang, Bo; Jiang, Xiangrui
Journal: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2023; Vol. 253, Issue , pp. -. DOI: 10.1016/j.ejmech.2023.115320
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Discovery of bipyridine amide derivatives targeting pRXR?-PLK1 interaction for anticancer therapy
Author: Chen, Jun; Zhao, Taige; He, Fengming; Zhong, Yijing; Wang, Susu; Tang, Ziqing; Qiu, Yingkun; Wu, Zhen; Fang, Meijuan
Journal: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2023; Vol. 254, Issue , pp. -. DOI: 10.1016/j.ejmech.2023.115341
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Discovery of novel sulfonamide chromone-oxime derivatives as potent indoleamine 2,3-dioxygenase 1 inhibitors
Author: Wang, Ke; Song, Long-Hao; Liang, Qiao-Ling; Zhang, Ye; Ma, Xian-Li; Wang, Qi; Zhang, Hui-Yong; Jiang, Cai-Na; Wei, Jian-Hua; Huang, Ri-Zhen
Journal: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2023; Vol. 254, Issue , pp. -. DOI: 10.1016/j.ejmech.2023.115349
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Discovery of 7H-Pyrrolo[2,3-d]pyrimidine Derivatives as potent hematopoietic progenitor kinase 1 (HPK1) inhibitors
Author: Wu, Feifei; Li, Huiyu; An, Qi; Sun, Yaoliang; Yu, Jinghua; Cao, Wenting; Sun, Pu; Diao, Xingxing; Meng, Linghua; Xu, Shilin
Journal: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2023; Vol. 254, Issue , pp. -. DOI: 10.1016/j.ejmech.2023.115355
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1-Benzyloxy-5-phenyltetrazole derivatives highly active against androgen receptor-dependent prostate cancer cells
Author: Zhao, Shiting; Ali, Abdelsalam S.; Kong, Xinyu; Zhang, Yan; Liu, Xiaomin; Skidmore, Melissa A.; Forsyth, Craig M.; Paul, G.; Wu, Donghai; Xu, Yong; Francis, Craig L.
Journal: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2023; Vol. 246, Issue , pp. -. DOI: 10.1016/j.ejmech.2022.114982
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Synthesis and bioactivity evaluation of ferrocene-based hydroxamic acids as selective histone deacetylase 6 inhibitors
Author: Yan, Jiangkun; Yue, Kairui; Fan, Xuejing; Xu, Ximing; Wang, Jing; Qin, Mengting; Zhang, Qianer; Hou, Xiaohan; Li, Xiaoyang; Wang, Yong
Journal: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2023; Vol. 246, Issue , pp. -. DOI: 10.1016/j.ejmech.2022.115004
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Discovery of cysteine-targeting covalent histone methyltransferase inhibitors
Author: Zhao, Yifan; Jiang, Bo; Gu, Zhouyang; Chen, Tianle; Yu, Wei; Liu, Shiyin; Liu, Xing; Chen, Dongyin; Li, Fei; Chen, Weilin
Journal: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2023; Vol. 246, Issue , pp. -. DOI: 10.1016/j.ejmech.2022.115028
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A comprehensive overview of Artemisinin and its derivatives as anticancer agents
Author: Zeng, Zi-wei; Chen, Di; Chen, Lei; He, Bin; Li, Yan
Journal: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2023; Vol. 247, Issue , pp. -. DOI: 10.1016/j.ejmech.2022.115000
