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Design, Synthesis, and Insecticidal Evaluation of New Benzoylureas Containing Carbamate Groups Based on the Bipartite Model of Sulfonylurea Receptor Binding Site
Author: Zhang, Jingjing; Zhu, Hualing; Xiong, Lixia; Shi, Jun; Huang, Zhiqiang
Journal: LETTERS IN DRUG DESIGN & DISCOVERY. 2023; Vol. 20, Issue 1, pp. 110-118. DOI: 10.2174/1570180819666220512182621
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Design, Synthesis, and Anti-Bacterial Evaluation of Tetrahydrobenzothiophene Derivatives as Lipopolysaccharide Biogenesis Inhibitors
Author: Pei, Shuchen; Yang, Jinhua; Xia, Shihao; Tang, Shuting; Yuan, Kangyao; Chen, Jun
Journal: LETTERS IN DRUG DESIGN & DISCOVERY. 2023; Vol. 20, Issue 3, pp. 335-342. DOI: 10.2174/1570180819666220317151208
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Molecular Mechanism of Qingchang Suppository in the Treatment of Ulcerative Colitis Based on Network Pharmacology
Author: Lin, Zhancheng; Lu, Lu; Zhu, Lingyu
Journal: LETTERS IN DRUG DESIGN & DISCOVERY. 2023; Vol. 20, Issue 1, pp. 71-76. DOI: 10.2174/1570180819666220509070003
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Synthesis and Preliminary Biological Evaluation of New Phthalazinone Derivatives with PARP-1 and Cholinesterase Inhibitory Activities
Author: Lin, Yu; Gao, Chengzhi; Wang, Zhuyong; Zhang, Ruifeng; Chen, Yajun; Min, Zhenli
Journal: LETTERS IN DRUG DESIGN & DISCOVERY. 2023; Vol. 20, Issue 1, pp. 56-70. DOI: 10.2174/1570180819666220531144809
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Oxymatrine-induced Apoptosis in Fibroblasts like Synoviocytes via Regulation of miR-146a/TRAF6/JNK1 Axis in Rheumatoid Arthritis
Author: Li, Jing; Hong, Hua
Journal: LETTERS IN DRUG DESIGN & DISCOVERY. 2023; Vol. 20, Issue 2, pp. 232-237. DOI: 10.2174/1570180819666220530143250
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Design and Screening of KLHL22 Inhibitors by Homology Modeling, Molecular Docking, and Molecular Dynamics Simulation
Author: Gao, Chenglong; Sun, Chuance; Zhang, Lichuan; Zhang, Haoran; Yu, Rilei; Kang, Congmin
Journal: LETTERS IN DRUG DESIGN & DISCOVERY. 2023; Vol. 20, Issue 3, pp. 291-303. DOI: 10.2174/1570180819666220422101618