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Design, synthesis and biological evaluation of novel 3,4-dihydro-2H-[1,4] oxazino [2,3-f]quinazolin derivatives as EGFR-TKIs
Author: Qin, Xuemei; Liu, Peng; Li, Yihai; Hu, Liming; Liao, Yexin; Cao, Tingting; Yang, Lifang
Journal: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2023; Vol. 80, Issue , pp. -. DOI: 10.1016/j.bmcl.2022.129104
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A new class of CYP1B1 inhibitors derived from bentranil
Author: Yi, Lan; Huang, Xinyue; Yang, Meixian; Cai, Jiajing; Jia, Jianhua; Peng, Zhiping; Zhao, Zhenghuan; Yang, Fengyuan; Qiu, Dachuan
Journal: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2023; Vol. 80, Issue , pp. -. DOI: 10.1016/j.bmcl.2022.129112
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Trienomycin A-simplified analogs: Synthesis and anti-neuroinflammatory activity
Author: Luo, Yu-Qing; Bian, Zhao-Yuan; Xu, Dan-Dan; Tang, Jiang-Jiang; Gao, Jin-Ming
Journal: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2023; Vol. 80, Issue , pp. -. DOI: 10.1016/j.bmcl.2022.129122
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New cycloalkyl[b]thiophenylnicotinamide-based alpha-glucosidase inhibitors as promising anti-diabetic agents: Synthesis, in silico study, in vitro and in vivo evaluations
Author: Wang, Kai-Ming; Ge, Yong-Xi; Zhang, Jie; Chen, Yi-Tong; Zhang, Nai-Yu; Gu, Jin-Song; Fang, Lei; Zhang, Xin-Lei; Zhang, Juan; Jiang, Cheng-Shi
Journal: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2023; Vol. 79, Issue , pp. -. DOI: 10.1016/j.bmcl.2022.129069
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Accumulation of lankamycin derivative with a branched-chain sugar from a blocked mutant of chalcose biosynthesis in Streptomyces rochei 7434AN4
Author: Zhang, Mingge; Shuang, Bao; Arakawa, Kenji
Journal: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2023; Vol. 80, Issue , pp. -. DOI: 10.1016/j.bmcl.2023.129125
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Role of symmetry in 3,3-diphenyl-1,3-dihydroindol-2-one derivatives as inhibitors of translation initiation
Author: Yang, Hongwei; Chen, Ting; Denoyelle, Severine; Chen, Limo; Fan, Jing; Zhang, Yingzhen; Halperin, Jose A.; Chorev, Michael; Aktas, Bertal H.
Journal: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2023; Vol. 80, Issue , pp. -. DOI: 10.1016/j.bmcl.2022.129119
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Synthesis and antibacterial activity of novel 2-fluoro ketolide antibiotics with 11,12-quinoylalkyl side chains
Author: Jin, Longlong; Zhang, Xiaoxi; Luo, Zhigang; Wu, Xianfu; Zhao, Zhehui
Journal: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2023; Vol. 80, Issue , pp. -. DOI: 10.1016/j.bmcl.2022.129115
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Synthesis of pyrrolo[3,2-d]pyrimidineone derivatives as novel FXa inhibitors
Author: Yang, Jiabin; Su, Bolang; Liao, Ruizhu; Wang, Jinrui; Bo, Shuyu
Journal: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2023; Vol. 80, Issue , pp. -. DOI: 10.1016/j.bmcl.2023.129127
